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@ARTICLE{Ramp:1007355,
author = {Ramp, Paul and Mack, Christina and Wirtz, Astrid and Bott,
Michael},
title = {{A}lternative routes for production of the drug candidate
d-chiro-inositol with {C}orynebacterium glutamicum using
endogenous or promiscuous plant enzymes},
journal = {Metabolic engineering},
volume = {78},
issn = {1096-7176},
address = {Orlando, Fla.},
publisher = {Academic Press},
reportid = {FZJ-2023-02024},
pages = {1 - 10},
year = {2023},
note = {Biotechnologie 1},
abstract = {d-chiro-Inositol (DCI) is a promising drug candidate for
treating insulin resistance and associated diseases such as
type 2 diabetes or polycystic ovary syndrome. In this study,
we developed two production processes for DCI using
Corynebacterium glutamicum as host. In the first process,
myo-inositol (MI) is oxidized to 2-keto-myo-inositol (2KMI)
by the inositol dehydrogenase (IDH) IolG and then isomerized
to 1-keto-d-chiro-inositol (1KDCI) by the isomerases Cg0212
or Cg2312, both of which were identified in this work. 1KDCI
is then reduced to DCI by IolG. Overproduction of IolG and
Cg0212 in a chassis strain unable to degrade inositols
allowed the production of 1.1 g/L DCI from 10 g/L MI. As
both reactions involved are reversible, only a partial
conversion of MI to DCI can be achieved. To enable higher
conversion ratios, a novel route towards DCI was established
by utilizing the promiscuous activity of two plant-derived
enzymes, the NAD+-dependent d-ononitol dehydrogenase MtOEPa
and the NADPH-dependent d-pinitol dehydrogenase MtOEPb from
Medicago truncatula (barrelclover). Heterologous production
of these enzymes in the chassis strain led to the production
of 1.6 g/L DCI from 10 g/L MI. For replacing the substrate
MI by glucose, the two plant genes were co-expressed with
the endogenous myo-inositol-1-phosphate synthase gene ino1
either as a synthetic operon or using a novel, bicistronic
T7-based expression vector. With the single operon
construct, 0.75 g/L DCI was formed from 20 g/L glucose,
whereas with the bicistronic construct 1.2 g/L DCI was
obtained, disclosing C. glutamicum as an attractive host for
of d-chiro-inositol production.},
cin = {IBG-1},
ddc = {610},
cid = {I:(DE-Juel1)IBG-1-20101118},
pnm = {2171 - Biological and environmental resources for
sustainable use (POF4-217)},
pid = {G:(DE-HGF)POF4-2171},
typ = {PUB:(DE-HGF)16},
pubmed = {37146873},
UT = {WOS:001005297800001},
doi = {10.1016/j.ymben.2023.04.013},
url = {https://juser.fz-juelich.de/record/1007355},
}