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@ARTICLE{Khaled:1015354,
author = {Khaled, Mohammed and Rönnbäck, Isabel and Ilag, Leopold
L. and Gräslund, Astrid and Strodel, Birgit and Österlund,
Nicklas},
title = {{A} {H}airpin {M}otif in the {A}myloid-β {P}eptide {I}s
{I}mportant for {F}ormation of {D}isease-{R}elated
{O}ligomers},
journal = {Journal of the American Chemical Society},
volume = {145},
number = {33},
issn = {0002-7863},
address = {Washington, DC},
publisher = {ACS Publications},
reportid = {FZJ-2023-03674},
pages = {18340 - 18354},
year = {2023},
abstract = {The amyloid-β (Aβ) peptide is associated with the
development of Alzheimer’s disease and is known to form
highly neurotoxic prefibrillar oligomeric aggregates, which
are difficult to study due to their transient,
low-abundance, and heterogeneous nature. To obtain
high-resolution information about oligomer structure and
dynamics as well as relative populations of assembly states,
we here employ a combination of native ion mobility mass
spectrometry and molecular dynamics simulations. We find
that the formation of Aβ oligomers is dependent on the
presence of a specific β-hairpin motif in the peptide
sequence. Oligomers initially grow spherically but start to
form extended linear aggregates at oligomeric states larger
than those of the tetramer. The population of the extended
oligomers could be notably increased by introducing an
intramolecular disulfide bond, which prearranges the peptide
in the hairpin conformation, thereby promoting oligomeric
structures but preventing conversion into mature fibrils.
Conversely, truncating one of the β-strand-forming segments
of Aβ decreased the hairpin propensity of the peptide and
thus decreased the oligomer population, removed the
formation of extended oligomers entirely, and decreased the
aggregation propensity of the peptide. We thus propose that
the observed extended oligomer state is related to the
formation of an antiparallel sheet state, which then
nucleates into the amyloid state. These studies provide
increased mechanistic understanding of the earliest steps in
Aβ aggregation and suggest that inhibition of Aβ folding
into the hairpin conformation could be a viable strategy for
reducing the amount of toxic oligomers.},
cin = {IBI-7},
ddc = {540},
cid = {I:(DE-Juel1)IBI-7-20200312},
pnm = {5241 - Molecular Information Processing in Cellular Systems
(POF4-524)},
pid = {G:(DE-HGF)POF4-5241},
typ = {PUB:(DE-HGF)16},
pubmed = {37555670},
UT = {WOS:001044984100001},
doi = {10.1021/jacs.3c03980},
url = {https://juser.fz-juelich.de/record/1015354},
}