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@ARTICLE{Ismail:172163,
author = {Ismail, Shehab A and Chen, Yong-Xiang and Rusinova,
Alexandra and Chandra, Anchal and Bierbaum, Martin and
Gremer, Lothar and Triola, Gemma and Waldmann, Herbert and
Bastiaens, Philippe I H and Wittinghofer, Alfred},
title = {{A}rl2-{GTP} and {A}rl3-{GTP} regulate a {GDI}-like
transport system for farnesylated cargo},
journal = {Nature chemical biology},
volume = {7},
number = {12},
issn = {1552-4469},
address = {Basingstoke},
publisher = {Nature Publishing Group},
reportid = {FZJ-2014-05673},
pages = {942 - 949},
year = {2011},
abstract = {Lipidated Rho and Rab GTP-binding proteins are transported
between membranes in complex with solubilizing factors
called ‘guanine nucleotide dissociation inhibitors’
(GDIs). Unloading from GDIs using GDI displacement factors
(GDFs) has been proposed but remains mechanistically
elusive. PDEd is a putative solubilizing factor for several
prenylated Ras-subfamily proteins. Here we report the
structure of fully modified farnesylated Rheb-GDP in complex
with PDEd. The structure explains the nucleotide-independent
binding of Rheb to PDEd and the relaxed specificity of PDEd.
We demonstrate that the G proteins Arl2 and Arl3 act in a
GTP-dependent manner as allosteric release factors for
farnesylated cargo. We thus describe a new transport system
for farnesylated G proteins involving a GDI-like molecule
and an unequivocal GDF. Considering the importance of PDEd
for proper Ras and Rheb signaling, this study is
instrumental in developing a new target for anticancer
therapy.},
cin = {ICS-6},
ddc = {540},
cid = {I:(DE-Juel1)ICS-6-20110106},
pnm = {452 - Structural Biology (POF2-452)},
pid = {G:(DE-HGF)POF2-452},
typ = {PUB:(DE-HGF)16},
UT = {WOS:000297166200018},
pubmed = {pmid:22002721},
doi = {10.1038/nchembio.686},
url = {https://juser.fz-juelich.de/record/172163},
}