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@ARTICLE{Quy:186054,
author = {Quy, Vo and Carnevale, Vincenzo and Manganaro, Lara and
Lusic, Marina and Rossetti, Giulia and Leone, Vanessa and
Fenollar-Ferrer, Cristina and Raugei, Simone and Sal,
Giannino and Giacca, Mauro and Carloni, Paolo},
title = {{HIV}-1 {I}ntegrase {B}inding to its {C}ellular {P}artners:
{A} {P}erspective from {C}omputational {B}iology},
journal = {Current pharmaceutical design},
volume = {20},
number = {21},
issn = {1381-6128},
address = {Hilversum},
publisher = {Bentham Science Publ.},
reportid = {FZJ-2015-00155},
pages = {3412 - 3421},
year = {2014},
abstract = {Viral DNA integration into the infected cell genome is an
essential step in the HIV-1 life cycle. Hence, the viral
integrase enzyme has become an important target for
antiviral therapy. The integrase's activity action relies on
the binding to its cellular partners, therefore the
knowledge of the structural determinants is very important
from a therapeutic perspective. Here we first review
published computer-aided structural predictions of HIV-1
integrase in complex with its interactors. These include DNA
and the human HAT protein. Next, we present a prediction of
the complex between HIV-1 integrase with the human
prolyl-isomerase-1 (hPin1) enzyme. Interaction with hPin1 is
crucial for efficient HIV-1 infection and it increases
integrase stability (Manganaro et. al 2010, Nat. Med. 16,
329). The modeling presented here, which is validated
against experimental data, provides a rationale for a
variety of viral protein's mutations which impair protein
function and HIV-1 virus replication in vivo without
significantly affecting enzymatic activity.},
cin = {JSC / IAS-5 / INM-9},
ddc = {610},
cid = {I:(DE-Juel1)JSC-20090406 / I:(DE-Juel1)IAS-5-20120330 /
I:(DE-Juel1)INM-9-20140121},
pnm = {411 - Computational Science and Mathematical Methods
(POF2-411)},
pid = {G:(DE-HGF)POF2-411},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:24001231},
UT = {WOS:000337899300004},
doi = {10.2174/13816128113199990631},
url = {https://juser.fz-juelich.de/record/186054},
}