% IMPORTANT: The following is UTF-8 encoded. This means that in the presence
% of non-ASCII characters, it will not work with BibTeX 0.99 or older.
% Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or
% “biber”.
@ARTICLE{Dibenedetto:201097,
author = {Dibenedetto, Domenica and Rossetti, Giulia and Caliandro,
Rocco and Carloni, Paolo},
title = {{A} {M}olecular {D}ynamics {S}imulation-{B}ased
{I}nterpretation of {N}uclear {M}agnetic {R}esonance
{M}ultidimensional {H}eteronuclear {S}pectra of
α-{S}ynuclein·{D}opamine {A}dducts},
journal = {Biochemistry},
volume = {52},
number = {38},
issn = {1520-4995},
address = {Columbus, Ohio},
publisher = {American Chemical Society},
reportid = {FZJ-2015-03402},
pages = {6672 - 6683},
year = {2013},
abstract = {Multidimensional heteronuclear nuclear magnetic resonance
(NMR) spectroscopy provides valuable structural information
about adducts between naturally unfolded proteins and their
ligands. These are often highly pharmacologically relevant.
Unfortunately, the determination of the contributions to
observed chemical shifts changes upon ligand binding is
complicated. Here we present a tool that uses molecular
dynamics (MD) trajectories to help interpret two-dimensional
(2D) NMR data. We apply this tool to the naturally unfolded
protein human α-synuclein interacting with dopamine, an
inhibitor of fibril formation, and with its oxidation
products in water solutions. By coupling 2D NMR experiments
with MD simulations of the adducts in explicit water, the
tool confirms with experimental data that the ligands bind
preferentially to 125YEMPS129 residues in the C-terminal
region and to a few residues of the so-called NAC region
consistently. It also suggests that the ligands might cause
conformational rearrangements of distal residues located at
the N-terminus. Hence, the performed analysis provides a
rationale for the observed changes in chemical shifts in
terms of direct contacts with the ligand and conformational
changes in the protein.},
cin = {IAS-5 / JSC / GRS},
ddc = {570},
cid = {I:(DE-Juel1)IAS-5-20120330 / I:(DE-Juel1)JSC-20090406 /
I:(DE-Juel1)GRS-20100316},
pnm = {411 - Computational Science and Mathematical Methods
(POF2-411)},
pid = {G:(DE-HGF)POF2-411},
typ = {PUB:(DE-HGF)16},
UT = {WOS:000330099300011},
pubmed = {pmid:23964651},
doi = {10.1021/bi400367r},
url = {https://juser.fz-juelich.de/record/201097},
}