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@ARTICLE{Stoll:29865,
      author       = {Stoll, T. and Ermert, J. and Oya, S. and Kung, H. F. and
                      Coenen, H. H.},
      title        = {{A}pplication of n.c.a. 4-[18{F}]fluorophenol in diaryl
                      ether syntheses of 2-(4-[18{F}]fluorophenoxy)-benzylamines},
      journal      = {Journal of labelled compounds and radiopharmaceuticals},
      volume       = {47},
      number       = {7},
      issn         = {0362-4803},
      address      = {New York, NY [u.a.]},
      publisher    = {Wiley},
      reportid     = {PreJuSER-29865},
      pages        = {443 - 455},
      year         = {2004},
      note         = {Record converted from VDB: 12.11.2012},
      abstract     = {The availability of no-carrier-added (n.c.a.)
                      4-[F-18]fluorophenol offers the possibility of introducing
                      the 4-[F-18]fluorophenoxy moiety into potential
                      radiopharmaceuticals. Besides alkyl-aryl ether synthesis
                      using n.c.a. 4-[F-18]fluorophenol the diaryl ether coupling
                      is an attractive synthetic method to enlarge the spectrum of
                      interesting labelling procedures. As examples the syntheses
                      of n.c.a. 2-(4-[F-18]fluorophenoxy)-N,N-dimethylbenzylamine
                      and n.c.a. 2-(4-[F-18]fluorophenoxy)-N-methylbenzylamine
                      were realized by an Ullmann ether synthesis of corresponding
                      2-bromobenzoic acid amides using
                      tetrakis(acetonitrile)copper(I) hexafluorophosphate as
                      catalyst and a subsequent reduction of the amides formed.
                      The radiochemical yield of the coupling varied between 5 and
                      $65\%$ based on labelled 4-[F-18]fluorophenol. Both
                      compounds are structural analogues of recently published
                      radiotracers for imaging the serotonin reuptake transporter
                      sites (SERT). However, in vitro binding assays of both
                      molecules showed only a low affinity towards monoamine
                      transporters. Copyright (C) 2004 John Wiley Sons, Ltd.},
      keywords     = {J (WoSType)},
      cin          = {INC},
      ddc          = {540},
      cid          = {I:(DE-Juel1)VDB53},
      pnm          = {Neurowissenschaften},
      pid          = {G:(DE-Juel1)FUEK255},
      shelfmark    = {Biochemical Research Methods / Chemistry, Medicinal /
                      Chemistry, Analytical / Pharmacology $\&$ Pharmacy},
      typ          = {PUB:(DE-HGF)16},
      UT           = {WOS:000222499000006},
      doi          = {10.1002/jlcr.828},
      url          = {https://juser.fz-juelich.de/record/29865},
}