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000825304 1001_ $$0P:(DE-Juel1)169356$$aKrapf, Philipp$$b0$$ufzj
000825304 245__ $$aSeyferth-Gilbert Homologation as a Route to 18 F-Labeled Building Blocks: Preparation of Radiofluor­inated Phenylacetylenes and Their Application in PET Chemistry
000825304 260__ $$aWeinheim$$bWiley-VCH Verl.$$c2016
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000825304 520__ $$aA convenient method for the preparation of hitherto unknown ([F-18]fluorophenyl)acetylenes ([F-18]FPAs) using the Seyferth-Gilbert homologation is reported. The novel building blocks were efficiently prepared from easily accessible [F-18]fluorobenzaldehydes by using the Bestmann-Ohira reagent. High radiochemical yields and excellent radiochemical purities were achieved within only 20 min of reaction time; 2- and 4-[F-18]FPAs were applied to prepare radiofluorinated heterocycles by using different cycloaddition and cross-coupling reactions. Additionally, these building blocks were used to prepare three novel PET tracers. Thus, an artificial radiofluorinated protected amino acid [F-18]10, a COX-2-specific ligand [F-18]14, and a PSMA-selective inhibitor [F-18]16 were obtained in high radiochemical yields.
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000825304 7001_ $$0P:(DE-Juel1)169321$$aRicharz, Raphael$$b1$$ufzj
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000825304 7001_ $$0P:(DE-Juel1)166419$$aNeumaier, Bernd$$b3$$eCorresponding author$$ufzj
000825304 7001_ $$0P:(DE-HGF)0$$aZlatopolskiy, Boris D.$$b4
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