000828196 001__ 828196 000828196 005__ 20220930130118.0 000828196 0247_ $$2doi$$a10.1002/chem.201604633 000828196 0247_ $$2ISSN$$a0947-6539 000828196 0247_ $$2ISSN$$a1521-3765 000828196 0247_ $$2WOS$$aWOS:000395775700003 000828196 0247_ $$2altmetric$$aaltmetric:15566668 000828196 0247_ $$2pmid$$apmid:27943464 000828196 037__ $$aFZJ-2017-02164 000828196 082__ $$a540 000828196 1001_ $$0P:(DE-Juel1)166483$$aZischler, Johannes$$b0 000828196 245__ $$aAlcohol-Enhanced Cu-Mediated Radiofluorination 000828196 260__ $$aWeinheim$$bWiley-VCH$$c2017 000828196 3367_ $$2DRIVER$$aarticle 000828196 3367_ $$2DataCite$$aOutput Types/Journal article 000828196 3367_ $$0PUB:(DE-HGF)16$$2PUB:(DE-HGF)$$aJournal Article$$bjournal$$mjournal$$s1490680069_14621 000828196 3367_ $$2BibTeX$$aARTICLE 000828196 3367_ $$2ORCID$$aJOURNAL_ARTICLE 000828196 3367_ $$00$$2EndNote$$aJournal Article 000828196 520__ $$aThe potential of many 18F-labeled (hetero)aromatics for applications in positron emission tomography remains underexplored because convenient procedures for their radiosynthesis are lacking. Consequently, simple methods to prepare radiofluorinated (hetero)arenes are highly sought after. Herein, we report the beneficial effect of primary and secondary alcohols on Cu-mediated 18F-labeling. This observation contradicts the assumption that such alcohols are inappropriate solvents for aromatic fluorination. Therefore, we developed a protocol for rapid radiolabeling of an extraordinarily broad scope of boronic and stannyl substrates under general reaction conditions. Notably, radiofluorinated indoles, phenols, and anilines were synthesized directly from the corresponding unprotected precursors. Furthermore, the novel method enabled the preparation of radiofluorinated tryptophans, [18F]F-DPA, [18F]DAA1106, 6-[18F]FDA, and 6-[18F]FDOPA 000828196 536__ $$0G:(DE-HGF)POF3-573$$a573 - Neuroimaging (POF3-573)$$cPOF3-573$$fPOF III$$x0 000828196 588__ $$aDataset connected to CrossRef 000828196 7001_ $$0P:(DE-HGF)0$$aKolks, Niklas$$b1 000828196 7001_ $$0P:(DE-Juel1)162416$$aModemann, Daniel$$b2$$ufzj 000828196 7001_ $$0P:(DE-Juel1)166419$$aNeumaier, Bernd$$b3$$eCorresponding author 000828196 7001_ $$0P:(DE-HGF)0$$aZlatopolskiy, Boris D.$$b4 000828196 773__ $$0PERI:(DE-600)1478547-x$$a10.1002/chem.201604633$$gVol. 23, no. 14, p. 3251 - 3256$$n14$$p3251 - 3256$$tChemistry - a European journal$$v23$$x0947-6539$$y2017 000828196 8767_ $$92017-03-30$$d2017-04-18$$eCover$$jZahlung erfolgt$$p201604633$$zFront cover 000828196 909CO $$ooai:juser.fz-juelich.de:828196$$pOpenAPC$$pVDB$$popenCost 000828196 9101_ $$0I:(DE-588b)5008462-8$$6P:(DE-Juel1)166483$$aForschungszentrum Jülich$$b0$$kFZJ 000828196 9101_ $$0I:(DE-588b)5008462-8$$6P:(DE-Juel1)162416$$aForschungszentrum Jülich$$b2$$kFZJ 000828196 9101_ $$0I:(DE-588b)5008462-8$$6P:(DE-Juel1)166419$$aForschungszentrum Jülich$$b3$$kFZJ 000828196 9131_ $$0G:(DE-HGF)POF3-573$$1G:(DE-HGF)POF3-570$$2G:(DE-HGF)POF3-500$$3G:(DE-HGF)POF3$$4G:(DE-HGF)POF$$aDE-HGF$$bKey Technologies$$lDecoding the Human Brain$$vNeuroimaging$$x0 000828196 9141_ $$y2017 000828196 915__ $$0StatID:(DE-HGF)0420$$2StatID$$aNationallizenz 000828196 915__ $$0StatID:(DE-HGF)0200$$2StatID$$aDBCoverage$$bSCOPUS 000828196 915__ $$0StatID:(DE-HGF)0300$$2StatID$$aDBCoverage$$bMedline 000828196 915__ $$0StatID:(DE-HGF)0310$$2StatID$$aDBCoverage$$bNCBI Molecular Biology Database 000828196 915__ $$0StatID:(DE-HGF)0100$$2StatID$$aJCR$$bCHEM-EUR J : 2015 000828196 915__ $$0StatID:(DE-HGF)0199$$2StatID$$aDBCoverage$$bThomson Reuters Master Journal List 000828196 915__ $$0StatID:(DE-HGF)0110$$2StatID$$aWoS$$bScience Citation Index 000828196 915__ $$0StatID:(DE-HGF)0150$$2StatID$$aDBCoverage$$bWeb of Science Core Collection 000828196 915__ $$0StatID:(DE-HGF)0111$$2StatID$$aWoS$$bScience Citation Index Expanded 000828196 915__ $$0StatID:(DE-HGF)1150$$2StatID$$aDBCoverage$$bCurrent Contents - Physical, Chemical and Earth Sciences 000828196 915__ $$0StatID:(DE-HGF)9905$$2StatID$$aIF >= 5$$bCHEM-EUR J : 2015 000828196 920__ $$lyes 000828196 9201_ $$0I:(DE-Juel1)INM-5-20090406$$kINM-5$$lNuklearchemie$$x0 000828196 980__ $$ajournal 000828196 980__ $$aVDB 000828196 980__ $$aI:(DE-Juel1)INM-5-20090406 000828196 980__ $$aUNRESTRICTED 000828196 980__ $$aAPC