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@ARTICLE{Zischler:828196,
      author       = {Zischler, Johannes and Kolks, Niklas and Modemann, Daniel
                      and Neumaier, Bernd and Zlatopolskiy, Boris D.},
      title        = {{A}lcohol-{E}nhanced {C}u-{M}ediated {R}adiofluorination},
      journal      = {Chemistry - a European journal},
      volume       = {23},
      number       = {14},
      issn         = {0947-6539},
      address      = {Weinheim},
      publisher    = {Wiley-VCH},
      reportid     = {FZJ-2017-02164},
      pages        = {3251 - 3256},
      year         = {2017},
      abstract     = {The potential of many 18F-labeled (hetero)aromatics for
                      applications in positron emission tomography remains
                      underexplored because convenient procedures for their
                      radiosynthesis are lacking. Consequently, simple methods to
                      prepare radiofluorinated (hetero)arenes are highly sought
                      after. Herein, we report the beneficial effect of primary
                      and secondary alcohols on Cu-mediated 18F-labeling. This
                      observation contradicts the assumption that such alcohols
                      are inappropriate solvents for aromatic fluorination.
                      Therefore, we developed a protocol for rapid radiolabeling
                      of an extraordinarily broad scope of boronic and stannyl
                      substrates under general reaction conditions. Notably,
                      radiofluorinated indoles, phenols, and anilines were
                      synthesized directly from the corresponding unprotected
                      precursors. Furthermore, the novel method enabled the
                      preparation of radiofluorinated tryptophans, [18F]F-DPA,
                      [18F]DAA1106, 6-[18F]FDA, and 6-[18F]FDOPA},
      cin          = {INM-5},
      ddc          = {540},
      cid          = {I:(DE-Juel1)INM-5-20090406},
      pnm          = {573 - Neuroimaging (POF3-573)},
      pid          = {G:(DE-HGF)POF3-573},
      typ          = {PUB:(DE-HGF)16},
      UT           = {WOS:000395775700003},
      pubmed       = {pmid:27943464},
      doi          = {10.1002/chem.201604633},
      url          = {https://juser.fz-juelich.de/record/828196},
}