% IMPORTANT: The following is UTF-8 encoded. This means that in the presence % of non-ASCII characters, it will not work with BibTeX 0.99 or older. % Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or % “biber”. @ARTICLE{Palermo:829379, author = {Palermo, Giulia and Minniti, Elirosa and Greco, Maria Laura and Riccardi, Laura and Simoni, Elena and Convertino, Marino and Marchetti, Chiara and Rosini, Michela and Sissi, Claudia and Minarini, Anna and De Vivo, Marco}, title = {{A}n optimized polyamine moiety boosts the potency of human type {II} topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate {F}14512}, journal = {Chemical communications}, volume = {51}, number = {76}, issn = {1364-548X}, address = {Cambridge}, publisher = {Soc.}, reportid = {FZJ-2017-03092}, pages = {14310 - 14313}, year = {2015}, abstract = {Combined computational–experimental analyses explain and quantify the spermine-vectorized F14512's boosted potency as a topoII poison. We found that an optimized polyamine moiety boosts drug binding to the topoII/DNA cleavage complex, rather than to the DNA alone. These results provide new structural bases and key reference data for designing new human topoII poisons.}, cin = {IAS-5 / INM-9}, ddc = {540}, cid = {I:(DE-Juel1)IAS-5-20120330 / I:(DE-Juel1)INM-9-20140121}, pnm = {899 - ohne Topic (POF3-899)}, pid = {G:(DE-HGF)POF3-899}, typ = {PUB:(DE-HGF)16}, UT = {WOS:000361073400005}, pubmed = {pmid:26234198}, doi = {10.1039/C5CC05065K}, url = {https://juser.fz-juelich.de/record/829379}, }