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@ARTICLE{Amundarain:861855,
author = {Amundarain, María Julia and Ribeiro, Rui Pedro and
Costabel, Marcelo Daniel and Giorgetti, Alejandro},
title = {{GABA} {A} receptor family: overview on structural
characterization},
journal = {Future medicinal chemistry},
volume = {11},
number = {3},
issn = {1756-8927},
address = {London},
publisher = {Future Science},
reportid = {FZJ-2019-02276},
pages = {229 - 245},
year = {2019},
abstract = {The pentameric γ-aminobutyric acid type A receptors are
ion channels activated by ligands, which intervene in the
rapid inhibitory transmission in the mammalian CNS. Due to
their rich pharmacology and therapeutic potential, it is
essential to understand their structure and function
thoroughly. This deep characterization was hampered by the
lack of experimental structural information for many years.
Thus, computational techniques have been extensively
combined with experimental data, in order to undertake the
study of γ-aminobutyric acid type A receptors and their
interaction with drugs. Here, we review the exciting journey
made to assess the structures of these receptors and outline
major outcomes. Finally, we discuss the brand new structure
of the α1β2γ2 subtype and the amazing advances it brings
to the field.},
cin = {IAS-5 / INM-9},
ddc = {540},
cid = {I:(DE-Juel1)IAS-5-20120330 / I:(DE-Juel1)INM-9-20140121},
pnm = {574 - Theory, modelling and simulation (POF3-574)},
pid = {G:(DE-HGF)POF3-574},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:30801199},
UT = {WOS:000465356900007},
doi = {10.4155/fmc-2018-0336},
url = {https://juser.fz-juelich.de/record/861855},
}