% IMPORTANT: The following is UTF-8 encoded. This means that in the presence
% of non-ASCII characters, it will not work with BibTeX 0.99 or older.
% Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or
% “biber”.
@ARTICLE{Orlovskaya:864918,
author = {Orlovskaya, Victoriya V. and Modemann, Daniel and
Kutnetsova, Olga F. and Fedorova, Olga S. and Urusova,
Elizaveta and Kolks, Niklas and Neumaier, Bernd and
Krasikova, Raisa N. and Zlatopolskiy, Boris},
title = {{A}lcohol-{S}upported {C}u-{M}ediated 18{F}-{F}luorination
of {I}odonium {S}alts under “{M}inimalist” {C}onditions},
journal = {Molecules},
volume = {24},
number = {17},
issn = {1420-3049},
address = {Basel},
publisher = {MDPI},
reportid = {FZJ-2019-04521},
pages = {3197},
year = {2019},
abstract = {In the era of personalized precision medicine, positron
emission tomography (PET) and related hybrid methods like
PET/CT and PET/MRI gain recognition as indispensable tools
of clinical diagnostics. A broader implementation of these
imaging modalities in clinical routine is closely dependent
on the increased availability of established and emerging
PET-tracers, which in turn could be accessible by the
development of simple, reliable, and efficient radiolabeling
procedures. A further requirement is a cGMP production of
imaging probes in automated synthesis modules. Herein, a
novel protocol for the efficient preparation of 18F-labeled
aromatics via Cu-mediated radiofluorination of
(aryl)(mesityl)iodonium salts without the need of
evaporation steps is described. Labeled aromatics were
prepared in high radiochemical yields simply by heating of
iodonium [18F]fluorides with the Cu-mediator in methanolic
DMF. The iodonium [18F]fluorides were prepared by direct
elution of 18F− from an anion exchange resin with
solutions of the corresponding precursors in MeOH/DMF. The
practicality of the novel method was confirmed by the
racemization-free production of radiolabeled
fluorophenylalanines, including hitherto unknown
3-[18F]FPhe, in $22–69\%$ isolated radiochemical yields as
well as its direct implementation into a remote-controlled
synthesis unit.},
cin = {INM-5},
ddc = {540},
cid = {I:(DE-Juel1)INM-5-20090406},
pnm = {573 - Neuroimaging (POF3-573)},
pid = {G:(DE-HGF)POF3-573},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:31484375},
UT = {WOS:000488613700177},
doi = {10.3390/molecules24173197},
url = {https://juser.fz-juelich.de/record/864918},
}