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@ARTICLE{Rossetti:866070,
author = {Rossetti, Giulia and Kless, Achim and Lai, Luhua and
Outeiro, Tiago F. and Carloni, Paolo},
title = {{I}nvestigating targets for neuropharmacological
intervention by molecular dynamics simulations},
journal = {Biochemical Society transactions},
volume = {47},
number = {3},
issn = {1470-8752},
address = {London},
publisher = {Biochemical Society},
reportid = {FZJ-2019-05309},
pages = {909 - 918},
year = {2019},
abstract = {Medical research has identified over 500 brain disorders.
Among these, there are still only very few neuropathologies
whose causes are fully understood and, consequently, very
few drugs whose mechanism of action is known. No FDA drug
has been identified for major neurodegenerative diseases,
such as Alzheimer's and Parkinson's. We still lack effective
treatments and strategies for modulating progression or even
early neurodegenerative disease onset diagnostic tools. A
great support toward the highly needed identification of
neuroactive drugs comes from computer simulation methods
and, in particular, from molecular dynamics (MD). This
provides insight into structure–function relationship of a
target and predicts structure, dynamics and energetics of
ligand/target complexes under biologically relevant
conditions like temperature and physiological saline
concentration. Here, we present examples of the predictive
power of MD for neuroactive ligands/target complexes. This
brief survey from our own research shows the usefulness of
partnerships between academia and industry, and from joint
efforts between experimental and theoretical groups.},
cin = {IAS-5 / INM-9 / JSC},
ddc = {540},
cid = {I:(DE-Juel1)IAS-5-20120330 / I:(DE-Juel1)INM-9-20140121 /
I:(DE-Juel1)JSC-20090406},
pnm = {572 - (Dys-)function and Plasticity (POF3-572) / 511 -
Computational Science and Mathematical Methods (POF3-511)},
pid = {G:(DE-HGF)POF3-572 / G:(DE-HGF)POF3-511},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:31085614},
UT = {WOS:000473225600013},
doi = {10.1042/BST20190048},
url = {https://juser.fz-juelich.de/record/866070},
}