% IMPORTANT: The following is UTF-8 encoded. This means that in the presence
% of non-ASCII characters, it will not work with BibTeX 0.99 or older.
% Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or
% “biber”.
@ARTICLE{Altenburg:885465,
author = {Altenburg, Bianca and Frings, Marcus and Schöbel,
Jan-Hendrik and Goßen, Jonas and Pannen, Kristina and
Vanderliek, Kim and Rossetti, Giulia and Koschmieder,
Steffen and Chatain, Nicolas and Bolm, Carsten},
title = {{C}hiral {A}nalogues of {PFI}-1 as {BET} {I}nhibitors and
{T}heir {F}unctional {R}ole in {M}yeloid {M}alignancies},
journal = {ACS medicinal chemistry letters},
volume = {11},
number = {10},
issn = {1948-5875},
address = {Washington, DC},
publisher = {ACS},
reportid = {FZJ-2020-03848},
pages = {1928–1934},
year = {2020},
abstract = {Structural analogues of PFI-1 varying at the sulfur core
were prepared, and their activities as BET inhibitors in
myeloid cell lines and primary cells from patients with
acute myeloid leukemia were studied. Docking calculations
followed by molecular dynamics simulations revealed the
binding mode of the newly prepared inhibitors, suggesting
explanations for the observed high enantiospecificity of the
inhibitory activity.},
cin = {IAS-5 / INM-9 / JSC},
ddc = {610},
cid = {I:(DE-Juel1)IAS-5-20120330 / I:(DE-Juel1)INM-9-20140121 /
I:(DE-Juel1)JSC-20090406},
pnm = {573 - Neuroimaging (POF3-573) / 572 - (Dys-)function and
Plasticity (POF3-572) / 574 - Theory, modelling and
simulation (POF3-574) / 511 - Computational Science and
Mathematical Methods (POF3-511)},
pid = {G:(DE-HGF)POF3-573 / G:(DE-HGF)POF3-572 /
G:(DE-HGF)POF3-574 / G:(DE-HGF)POF3-511},
typ = {PUB:(DE-HGF)16},
pubmed = {33062175},
UT = {WOS:000580567800022},
doi = {10.1021/acsmedchemlett.9b00625},
url = {https://juser.fz-juelich.de/record/885465},
}