TY  - JOUR
AU  - Humpert, Swen
AU  - Omrane, Mohamed A.
AU  - Urusova, Elizaveta
AU  - Gremer, Lothar
AU  - Willbold, Dieter
AU  - Endepols, Heike
AU  - Krasikova, Raisa N.
AU  - Neumaier, Bernd
AU  - Zlatopolskiy, Boris D.
TI  - Rapid 18 F-labeling via Pd-catalyzed S -arylation in aqueous medium
JO  - Chemical communications
VL  - 57
SN  - 1364-548X
CY  - Cambridge
PB  - Soc.
M1  - FZJ-2021-01553
SP  - 3547-3550 
PY  - 2021
AB  - We report radiolabeling of thiol-containing substrates via Pd-catalyzed S-arylation with 2-[18F]fluoro-5-iodopyridine, which is readily accessible using the “minimalist” radiofluorination method. The practicality of the procedure was confirmed by preparation of a novel PSMA-specific PET-tracer as well as labeling of glutathione, Aβ oligomer-binding RD2 peptide, bovine serum albumin and PSMA I&S.
LB  - PUB:(DE-HGF)16
C6  - 33870341
UR  - <Go to ISI:>//WOS:000637899600020
DO  - DOI:10.1039/D1CC00745A
UR  - https://juser.fz-juelich.de/record/891479
ER  -