% IMPORTANT: The following is UTF-8 encoded. This means that in the presence % of non-ASCII characters, it will not work with BibTeX 0.99 or older. % Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or % “biber”. @ARTICLE{Koch:902967, author = {Koch, Katharina and Hartmann, Rudolf and Suwala, Abigail Kora and Rios, Dayana Herrera and Kamp, Marcel Alexander and Sabel, Michael and Steiger, Hans-Jakob and Willbold, Dieter and Sharma, Amit and Kahlert, Ulf Dietrich and Maciaczyk, Jarek}, title = {{O}verexpression of {C}ystine/{G}lutamate {A}ntiporter x{CT} {C}orrelates with {N}utrient {F}lexibility and {ZEB}1 {E}xpression in {H}ighly {C}lonogenic {G}lioblastoma {S}tem-like {C}ells ({GSC}s)}, journal = {Cancers}, volume = {13}, number = {23}, issn = {2072-6694}, address = {Basel}, publisher = {MDPI}, reportid = {FZJ-2021-04713}, pages = {6001 -}, year = {2021}, abstract = {Cancer stem-like cells mediate tumor initiation, progression, and therapy resistance; however, their identification and selective eradication remain challenging. Herein, we analyze the metabolic dependencies of glioblastoma stem-like cells (GSCs) with high-resolution proton nuclear magnetic resonance (1H-NMR) spectroscopy. We stratify our in vitro GSC models into two subtypes primarily based on their relative amount of glutamine in relationship to glutamate (Gln/Glu). Gln/GluHigh GSCs were found to be resistant to glutamine deprivation, whereas Gln/GluLow GSCs respond with significantly decreased in vitro clonogenicity and impaired cell growth. The starvation resistance appeared to be mediated by an increased expression of the glutamate/cystine antiporter SLC7A11/xCT and efficient cellular clearance of reactive oxygen species (ROS). Moreover, we were able to directly correlate xCT-dependent starvation resistance and high Gln/Glu ratios with in vitro clonogenicity, since targeted differentiation of GSCs with bone morphogenic protein 4 (BMP4) impaired xCT expression, decreased the Gln/Glu ratio, and restored the sensitivity to glutamine starvation. Moreover, significantly reduced levels of the oncometabolites lactate (Lac), phosphocholine (PC), total choline (tCho), myo-inositol (Myo-I), and glycine (Gly) were observed in differentiated GSCs. Furthermore, we found a strong association between high Gln/Glu ratios and increased expression of Zinc finger E-box-binding homeobox 1 (ZEB1) and xCT in primary GBM tumor tissues. Our analyses suggest that the inhibition of xCT represents a potential therapeutic target in glioblastoma; thus, we could further extend its importance in GSC biology and stress responses. We also propose that monitoring of the intracellular Gln/Glu ratio can be used to predict nutrient stress resistance.}, cin = {IBI-7}, ddc = {610}, cid = {I:(DE-Juel1)IBI-7-20200312}, pnm = {5244 - Information Processing in Neuronal Networks (POF4-524)}, pid = {G:(DE-HGF)POF4-5244}, typ = {PUB:(DE-HGF)16}, pubmed = {34885110}, UT = {WOS:000762087200001}, doi = {10.3390/cancers13236001}, url = {https://juser.fz-juelich.de/record/902967}, }