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@ARTICLE{Ahmad:909641,
author = {Ahmad, Katya and Rizzi, Andrea and Capelli, Riccardo and
Mandelli, Davide and Lyu, Wenping and Carloni, Paolo},
title = {{E}nhanced-{S}ampling {S}imulations for the {E}stimation of
{L}igand {B}inding {K}inetics: {C}urrent {S}tatus and
{P}erspective},
journal = {Frontiers in molecular biosciences},
volume = {9},
issn = {2296-889X},
address = {Lausanne},
publisher = {Frontiers},
reportid = {FZJ-2022-03312},
pages = {899805},
year = {2022},
abstract = {The dissociation rate (koff) associated with ligand
unbinding events from proteins is a parameter of fundamental
importance in drug design. Here we review recent major
advancements in molecular simulation methodologies for the
prediction of koff. Next, we discuss the impact of the
potential energy function models on the accuracy of
calculated koff values. Finally, we provide a perspective
from high-performance computing and machine learning which
might help improve such predictions.},
cin = {IAS-5 / INM-9},
ddc = {570},
cid = {I:(DE-Juel1)IAS-5-20120330 / I:(DE-Juel1)INM-9-20140121},
pnm = {1215 - Simulations, Theory, Optics, and Analytics (STOA)
(POF4-121) / HBP SGA3 - Human Brain Project Specific Grant
Agreement 3 (945539)},
pid = {G:(DE-HGF)POF4-1215 / G:(EU-Grant)945539},
typ = {PUB:(DE-HGF)16},
pubmed = {35755817},
UT = {WOS:000814363000001},
doi = {10.3389/fmolb.2022.899805},
url = {https://juser.fz-juelich.de/record/909641},
}