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@ARTICLE{Jiang:817980,
author = {Jiang, Nan and Frenzel, Daniel and Schartmann, Elena and
van Groen, Thomas and Kadish, Inga and Shah, N. J. and
Langen, Karl-Josef and Willbold, Dieter and Willuweit,
Antje},
title = {{B}lood-brain barrier penetration of an {A}β-targeted,
arginine-rich, d-enantiomeric peptide},
journal = {Biochimica et biophysica acta / Biomembranes},
volume = {1858},
number = {11},
issn = {0005-2736},
address = {Amsterdam},
publisher = {Elsevier},
reportid = {FZJ-2016-04556},
pages = {2717 - 2724},
year = {2016},
abstract = {The application of small peptides targeting amyloid beta
(Aβ) is one of many drug development strategies for the
treatment of Alzheimer's disease (AD). We have previously
identified several peptides consisting solely of
D-enantiomeric amino acid residues obtained from
mirror-image phage display selection, which bind to Aβ in
different assembly states and eliminate toxic Aβ
aggregates. Some of these D-peptides show both diagnostic
and therapeutic potential in vitro and in vivo. Here we have
analysed the similarity of the arginine-rich D-peptide D3 to
the arginine-rich motif (ARM) of the human immunodeficiency
virus type 1 transactivator of transcription (HIV-Tat)
protein, and examined its in vivo blood-brain barrier (BBB)
permeability using wild type mice and transgenic mouse
models of Alzheimer's disease. We are able to demonstrate
that D3 rapidly enters the brain where it can be found
associated with amyloid plaques suggesting a direct
penetration of BBB.},
cin = {INM-4 / ICS-6 / JARA-BRAIN},
ddc = {570},
cid = {I:(DE-Juel1)INM-4-20090406 / I:(DE-Juel1)ICS-6-20110106 /
$I:(DE-82)080010_20140620$},
pnm = {573 - Neuroimaging (POF3-573)},
pid = {G:(DE-HGF)POF3-573},
typ = {PUB:(DE-HGF)16},
UT = {WOS:000385318800016},
pubmed = {pmid:27423267},
doi = {10.1016/j.bbamem.2016.07.002},
url = {https://juser.fz-juelich.de/record/817980},
}