TY - JOUR
AU - Zlatopolskiy, Boris D.
AU - Zischler, Johannes
AU - Krapf, Philipp
AU - Richarz, Raphael
AU - Lauchner, Katharina
AU - Neumaier, Bernd
TI - Minimalist approach meets green chemistry: Synthesis of 18F-labeled (hetero)aromatics in pure ethanol
JO - Journal of labelled compounds and radiopharmaceuticals
VL - 62
IS - 8
SN - 0362-4803
CY - New York, NY [u.a.]
PB - Wiley
M1 - FZJ-2019-03789
SP - 404 - 410
PY - 2019
AB - The application of toxic solvents and additives is inevitable for most of the described protocols for 18F‐labeling. Herein, a novel “green” procedure for nucleophilic aromatic radiofluorination of highly activated (hetero)aromatic substrates in pure EtOH is described. Using this method a series of 18F‐labeled (hetero)arenes have been synthesized in radiochemical yields (RCYs) of up to 97%.
LB - PUB:(DE-HGF)16
C6 - pmid:31162691
UR - <Go to ISI:>//WOS:000475397300006
DO - DOI:10.1002/jlcr.3776
UR - https://juser.fz-juelich.de/record/863802
ER -