Journal Article

FZJ-2021-01553

http://join2-wiki.gsi.de/foswiki/pub/Main/Artwork/join2_logo100x88.png Rapid 18 F-labeling via Pd-catalyzed S -arylation in aqueous medium

Humpert, S.FZJ* ; Omrane, M. A. ; Urusova, E.FZJ* ; Gremer, L.FZJ* ; Willbold, D.FZJ* ; Endepols, H.FZJ* ; Krasikova, R. N. ; Neumaier, B. (Corresponding author)FZJ* ; Zlatopolskiy, B. D.

2021
Soc. Cambridge

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Please use a persistent id in citations: http://hdl.handle.net/2128/27898  doi:10.1039/D1CC00745A

Abstract: We report radiolabeling of thiol-containing substrates via Pd-catalyzed S-arylation with 2-[18F]fluoro-5-iodopyridine, which is readily accessible using the “minimalist” radiofluorination method. The practicality of the procedure was confirmed by preparation of a novel PSMA-specific PET-tracer as well as labeling of glutathione, Aβ oligomer-binding RD2 peptide, bovine serum albumin and PSMA I&S.

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Contributing Institute(s):

1. Nuklearchemie (INM-5)
2. Strukturbiochemie (IBI-7)

Research Program(s):

1. 525 - Decoding Brain Organization and Dysfunction (POF4-525) (POF4-525)

Appears in the scientific report 2021

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Database coverage:
; ; ; Allianz-Lizenz / DFG ; Chemical Reactions ; Clarivate Analytics Master Journal List ; Current Contents - Physical, Chemical and Earth Sciences ; Ebsco Academic Search ; Essential Science Indicators ; IF >= 5 ; Index Chemicus ; JCR ; National-Konsortium ; Nationallizenz ; SCOPUS ; Science Citation Index Expanded ; Web of Science Core Collection

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